Pitolisant
Product Specifications
CAS Number
362665-56-3
Synonyms
BF2.649, Tiprolisant
Target
Histamine Receptor
Applications
Neuronal Signaling
Additionnal Information
Pitolisant (BF2.649, Tiprolisant) is a potent, selective antagonist of the non-imidazole histamine H3 receptor, with a Ki value of 0.16 nM and an EC50 of 1.5 nM as an inverse agonist. It enhances the activity of histaminergic neurons, promoting vigilance and cognitive function. It is useful in research on wakefulness, memory deficits, and cognitive disorders.
Storage Conditions
2 years -20°C liquid
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