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Asenapine

Product Specifications

CAS Number

65576-45-6

Synonyms

Org 5222, HSDB8061

Target

5-HT Receptor

Applications

Neuronal Signaling

Molecular Formula

C17H16ClNO

Additionnal Information

Asenapine (Org 5222, HSDB8061) is a multi-target receptor antagonist. It acts as an antagonist of serotonin receptors with pKi values of 8.4-10.5, adrenoceptors with pKi values of 8.9-9.5, dopamine receptors with pKi values of 8.9-9.4 and histamine receptors with pKi values of 8.2-9.0.

Storage Conditions

2 years -20°C liquid

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