Welcome to GenPrice! Check out our latest updates.

Shopping Cart (0)

Your cart is empty

Add some products to get started!

Tazemetostat hydrobromide

Product Specifications

CAS Number

1467052-75-0

Synonyms

EPZ-6438 hydrobromide

Target

EZH1/2

Applications

Epigenetics

Molecular Formula

C34H44N4O4.BrH

Additionnal Information

Tazemetostat hydrobromide (EPZ-6438 hydrobromide) is a potent, selective, and orally available inhibitor of EZH2. It inhibits EZH2 with IC50 values of 11 and 16 nM in peptide assay and nucleosome assay, respectively. Tazemetostat hydrobromide also inhibits EZH1 with an IC50 of 392 nM.

Frequently Asked Questions

More Discoveries

Explore Other Products

Browse additional items from our catalog

Mouse Skor2 qPCR Primer Pair
QM76782S 200 Tests

Mouse Skor2 qPCR Primer Pair

Sign In for Pricing
View Details
(-) -3-O -Acetylcatechin
orb2281656 5 mg

(-) -3-O -Acetylcatechin

Sign In for Pricing
View Details
Recombinant Saccharomyces cerevisiae ATPase expression protein 1, mitochondrial (AEP1)
MBS1214368-01 0.02 mg (E-Coli)

Recombinant Saccharomyces cerevisiae ATPase expression protein 1, mitochondrial (AEP1)

Sign In for Pricing
View Details
Recombinant Saccharomyces cerevisiae ATPase expression protein 1, mitochondrial (AEP1)
MBS1214368-02 0.02 mg (Yeast)

Recombinant Saccharomyces cerevisiae ATPase expression protein 1, mitochondrial (AEP1)

Sign In for Pricing
View Details
Recombinant Saccharomyces cerevisiae ATPase expression protein 1, mitochondrial (AEP1)
MBS1214368-03 0.1 mg (E-Coli)

Recombinant Saccharomyces cerevisiae ATPase expression protein 1, mitochondrial (AEP1)

Sign In for Pricing
View Details
Recombinant Saccharomyces cerevisiae ATPase expression protein 1, mitochondrial (AEP1)
MBS1214368-04 0.1 mg (Yeast)

Recombinant Saccharomyces cerevisiae ATPase expression protein 1, mitochondrial (AEP1)

Sign In for Pricing
View Details