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DMB

Product Specifications

CAS Number

281209-71-0

Synonyms

GLP-1R agonist 2

Target

Glucagon Receptor

Applications

GPCR & G Protein

Molecular Formula

C13H15Cl2N3O2S

Additionnal Information

DMB (GLP-1R agonist 2, Compound 2) is an agonist of the GLP-1 receptor (GLP-1R) with a Ki of 13.25 μM. It activates GLP-1R by forming hydrogen bonds with the Tyr42, Cys71, and Ser84 residues. DMB attenuates transient focal cerebral ischemia injury and inhibits neuronal apoptosis induced by MCAO.

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