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Tilfrinib

Product Specifications

CAS Number

1600515-49-8

Molecular Formula

C17H13N3O

Additionnal Information

Tilfrinib (Compound 4f) is a potent and selective inhibitor of the tyrosine-protein kinase Brk/PTK6, with an IC50 of 3.15 nM. It demonstrates significant anti-proliferative activity against breast cancer cell lines MCF7, HS-578T, and BT-549.

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