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AZD0780

Product Specifications

CAS Number

2455427-91-3

Target

PCSK9

Applications

Metabolism

Molecular Formula

C20H20F2N6O2

Additionnal Information

AZD0780 (Laroprovstat, Pcsk9-IN-12) is an orally potent inhibitor of PCSK9 with a Kd value of <200 nM. It directly binds to PCSK9, blocks its function, and significantly reduces LDL cholesterol levels, making it useful for dyslipidemia research.

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