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CAN508

Product Specifications

CAS Number

140651-18-9

Target

CDK

Applications

Cell Cycle

Smiles

NC1=C (N=NC2=CC=C (O) C=C2) C (=N[NH]1) N

Molecular Formula

C9H10N6O

Additionnal Information

CAN508 is a potent, ATP-competitive CDK9/cyclin T1 inhibitor with an IC50 of 0.35 μM, exhibits a 38-fold selectivity for CDK9/cyclin T1 over other CDK/cyclin complexes.

Storage Conditions

3 years -20°C powder

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