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IBG1

Product Specifications

CAS Number

2684292-71-3

Synonyms

PROTAC BRD4 Degrader-19

Target

Epigenetic Reader Domain

Applications

Epigenetics

Molecular Formula

C44H38N8O5S2

Additionnal Information

IBG1 (PROTAC BRD4 Degrader-19) is a PROTAC-like degrader specifically targeting BET bromodomains with a DC50 of 0.15 nM for BRD4. It consists of the BET inhibitor JQ1 linked to E7820 and functions through CRL4-DCAF16.

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