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RMC-7977

Product Specifications

CAS Number

2765082-12-8

Target

Ras

Applications

Apoptosis

Molecular Formula

C47H60N8O6S

Additionnal Information

RMC-7977 is a potent, reversible, tri-complex oral inhibitor that selectively targets active (GTP-bound) forms of KRAS, HRAS, and NRAS, which exhibits broad-spectrum activity against both mutant and wild-type variants (a RASMULTI (ON) inhibitor) . It also exhibits significant anti-tumor efficacy in pancreatic ductal adenocarcinoma (PDAC) .
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