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Palazestrant

Product Specifications

CAS Number

2092925-89-6

Synonyms

OP-1250

Target

Estrogen/progestogen Receptor

Applications

Endocrinology & Hormones

Molecular Formula

C28H36FN3O

Additionnal Information

Palazestrant (OP-1250) is an orally bioavailable complete antagonist of estrogen receptor (ER) that blocks ER activity. It exhibits antiproliferative and antitumor activity in ER-positive (ER+) breast cancer models.
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