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Monlunabant

Product Specifications

CAS Number

2712480-46-9

Synonyms

INV-202, (S) -MRI-1891

Target

Cannabinoid Receptor

Applications

Neuronal Signaling

Molecular Formula

C26H22ClF3N6O3S

Additionnal Information

Monlunabant (INV-202, (S) -MRI-1891) is a peripherally acting inverse agonist of the cannabinoid type-1 receptor (CB1R), with the potential to treat respiratory and renal complications associated with metabolic disorders. It improves lung compliance in a mouse model of asthma and reduces renal fibrosis in a streptozotocin-induced diabetic nephropathy mouse model.

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