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Resigratinib

Product Specifications

CAS Number

2750709-91-0

Synonyms

KIN-3248

Target

FGFR

Applications

Protein Tyrosine Kinase

Molecular Formula

C26H27F2N7O3

Additionnal Information

Resigratinib (KIN-3248) is a potent, kinome selective, irreversible, orally bioavailable, small-molecule inhibitor of pan-FGFR. It exhibits dose-dependent tumor inhibition in FGFR driven cholangiocarcinoma, gastric, and bladder cancer xenograft models.

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