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AGI-24512

Product Specifications

CAS Number

2201066-53-5

Target

MAT2A

Applications

Methylation

Molecular Formula

C24H24N4O2

Additionnal Information

AGI-24512 is an inhibitor of MAT2A with an IC50 of 8 nM. It increases R-Loop formation and DNA damage in MTAP-deleted and WT cell models. It also exhibits anti-proliferative activity in vitro.
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