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Conteltinib (CT-707)

Product Specifications

CAS Number

1384860-29-0

Target

FAK

Applications

Protein Tyrosine Kinase

Molecular Formula

C32H45N9O3S

Additionnal Information

Conteltinib (CT-707) is a potent multikinase inhibitor of ALK, FAK, Pyk2, showing promising anti-tumor activities. Conteltinib exhibits significant inhibitory effects on FAK with an IC50 value of 1.6 nM in vitro kinase assay.

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