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HX531

Product Specifications

CAS Number

188844-34-0

Target

Retinoid Receptor

Applications

Metabolism

Molecular Formula

C29H29N3O4

Additionnal Information

HX531 is an orally active antagonist of RXR. HX531 enhances activation of the p53–p21Cip1 pathway and abrogates the anti-apoptotic effects of all-trans-retinoic acid (t-RA) . HX531 exhibits anti-obesity, anti-diabetic, and anti-melanoma properties.

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