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T025

Product Specifications

CAS Number

2407433-00-3

Target

CDK

Applications

Cell Cycle

Molecular Formula

C21H18N8

Additionnal Information

T025 is as an orally available and potent inhibitor of Cdc2‐like kinases (CLKs) with an IC50s of 0.93 nM, 1 nM, 14 nM, 1.5 nM for CLK1, CLK2, CLK3, DYRK1B respectively. It exhibits anti‐tumor efficacy and can be used in MYC‐driven cancer research.
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