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DN02

Product Specifications

Target

Epigenetic Reader Domain

Applications

Epigenetics

Molecular Formula

C22H24FN3O3

Additionnal Information

DN02 is a selective probe of BRD8 bromodomain family. It exhibits potency against BRD8 (1) with a Kd of 32 nM, and interestingly, demonstrated this activity to be selective over BRD8's second bromodomain (BRD8 (2) with a Kd of >1000 nM)

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