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AM-9747

Product Specifications

CAS Number

2691869-82-4

Synonyms

PRMT5-IN-25

Target

PRMT

Applications

Epigenetics

Molecular Formula

C24H21F3N6O

Additionnal Information

AM-9747 (PRMT5-IN-25) is a potent inhibitor of PRMT5 with a Ki of 0.06 nM. It exhibits antiproliferative activity and a significant oral antitumor effect in mouse models employing patient-derived xenografts (PDX) .

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