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MK-0159

Product Specifications

CAS Number

2641484-61-7

Synonyms

Compound 37

Target

CD markers

Applications

Transmembrane Transporters

Molecular Formula

C20H24N4O3S

Additionnal Information

MK-015 (Compound 37) is an inhibitor of CD38. MK-0159 inhibits human, mouse, and rat CD38 (cell-free assays) with IC50 values of 22, 3, and 70 nM, respectively. MK-0159 increases NAD+ (nicotinamide adenine dinucleotide) and reduces ADPR (adenosine diphosphate ribose) in whole blood and heart.

Storage Conditions

3 years -20°C powder

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