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Divarasib (GDC-6036)

Product Specifications

CAS Number

2417987-45-0

Synonyms

RG6330

Target

Ras

Applications

Apoptosis

Molecular Formula

C29H32ClF4N7O2

Additionnal Information

Divarasib (GDC-6036, RG6330) is a KRAS G12C inhibitor that binds irreversibly to switch II pocket of KRAS G12C (when in the inactive GDP-bound state) thereby blocking GTP binding and activation.

Storage Conditions

3 years -20°C powder

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