What is the catalog number for GA-017?

The catalog number for GA-017 is C01502-100mg.

What sizes are available for GA-017?

GA-017 is available in the following size(s): 100 mg.

GA-017 is currently made to order / not held in immediate stock. Contact us for lead time.

GA-017

Product Specifications

CAS Number

2351906-74-4

Target

LATS

Applications

Hippo

Smiles

CC\C (=N\NC (=O) NCC1=CC (=CC=C1) O) C2=C (O) C (=C (O) C=C2) C

Molecular Formula

C18H21N3O4

Additionnal Information

GA-017 inhibits the serine/threonine protein kinases large tumor suppressor kinase 1/2 (LATS1/2), which exerts inhibitory with IC50s against LATS1 and 2 of 4.10±0.79 and 3.92±0.42 nM, respectively, and competitively inhibits LATS1 and 2 against ATP, with Ki (inhibition constant) values of 0.58±0.11 and 0.25±0.03 nM, respectively.