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Lartesertib (M4076)

Product Specifications

CAS Number

2495096-26-7

Target

ATM/ATR

Applications

PI3K/Akt/mTOR

Molecular Formula

C23H21FN6O3

Additionnal Information

Lartesertib (M4076) inhibits Ataxia telangiectasia-mutated (ATM) kinase activity with a sub-nanomolar potency and shows remarkable selectivity against other protein kinases, suppresses DSB repair, clonogenic cancer cell growth, and potentiates antitumor activity of ionizing radiation in cancer cell lines.

Storage Conditions

3 years -20°C powder

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