CCT020312
Product Specifications
CAS Number
324759-76-4
Target
PERK
Applications
Apoptosis
Smiles
CCN (CC) CCC (=O) N1N=C (CC1C2=CC=C (Br) C=C2) C3=C (C4=CC=CC=C4) C5=C (NC3=O) C=CC (=C5) Br
Molecular Formula
C31H30Br2N4O2
Additionnal Information
CCT020312 is a selective PERK (EIF2AK3) activator with an EC50 of 5.1 μM. CCT020312 can be used for the selective activation of EIF2A-mediated translation control.
Storage Conditions
3 years -20°C powder
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