What is the catalog number for Masitinib mesylate?

The catalog number for Masitinib mesylate is C14688-100mg.

What sizes are available for Masitinib mesylate?

Masitinib mesylate is available in the following size(s): 100 mg.

Is Masitinib mesylate in stock?

Masitinib mesylate is currently made to order / not held in immediate stock. Contact us for lead time.

Masitinib mesylate

Product Specifications

CAS Number

1048007-93-7

Synonyms

AB-1010 mesylate

Target

C-Kit

Applications

Protein Tyrosine Kinase

Smiles

CN1CCN (CC1) CC2=CC=C (C=C2) C (=O) NC3=CC=C (C) C (=C3) NC4=NC (=CS4) C5=CN=CC=C5.C[S] (O) (=O) =O

Molecular Formula

C28H30N6OS.CH4O3S

Additionnal Information

Masitinib mesylate (AB-1010 mesylate) is a potent, orally bioavailable, and selective inhibitor of c-Kit with IC50 of 200 nM for human recombinant c-Kit, also inhibits PDGFRα/β with IC50s of 540/800 nM, Lyn with IC50 of 510 nM for LynB, and, to a lesser extent, FGFR3 and FAK.