Timapiprant Sodium
Product Specifications
CAS Number
950688-14-9
Synonyms
OC000459 sodium
Target
Prostaglandin Receptor
Applications
GPCR & G Protein
Smiles
[NaH].CC1=C (CC2=NC3=C (C=CC=C3) C=C2) C4=CC (=CC=C4[N]1CC (O) =O) F
Molecular Formula
C21H17FN2O2.Na
Additionnal Information
Timapiprant sodium (OC000459 sodium), a potent, selective, and orally active D prostanoid receptor 2 (DP2, also known as CRTH2) antagonist, potently displaces [3H]PGD2 from human recombinant DP2, rat recombinant DP2, and human native DP2 with Ki values of 13, 3 and 4 nM, respectively.
Storage Conditions
3 years -20°C powder
Frequently Asked Questions
More Discoveries
Explore Other Products
Browse additional items from our catalog