BMS-986122
Product Specifications
CAS Number
313669-88-4
Target
Opioid Receptor
Applications
Neuronal Signaling
Smiles
COC1=CC=C (C=C1Br) C2SCCN2[S] (=O) (=O) C3=CC=C (Cl) C=C3
Molecular Formula
C16H15BrClNO3S2
Additionnal Information
BMS-986122 is a selective, potent positive allosteric modulator of the mu-opioid receptor (μ-OR), shows potentiation of orthosteric agonist-mediated β-arrestin recruitment, adenylyl cyclase inhibition, and G protein activation, and potentiates DAMGO-mediated [35S]GTPγS binding in mouse brain membranes.
Storage Conditions
3 years -20°C powder
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