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IMP-1088

Product Specifications

CAS Number

2059148-82-0

Target

Others

Applications

Others

Molecular Formula

C25H29F2N5O

Additionnal Information

IMP-1088 is a potent dual inhibitor of human N-myristoyltransferases NMT1 and NMT2, with an IC50 of <1 nM for HsNMT1 and HsNMT2 and a Kd of <210 pM for HsNMT1. It effectively inhibits the production of infectious rhinovirus virions by blocking the N-myristoylation of the rhinovirus VP0 protein.

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