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Evocalcet

Product Specifications

CAS Number

870964-67-3

Synonyms

KHK7580

Target

CaSR

Applications

GPCR & G Protein

Molecular Formula

C24H26N2O2

Additionnal Information

Evocalcet (KHK7580) is an novel oral calcimimetic agent which acts via allosteric activation of the calcium sensing receptor (CaSR) . Evocalcet (0, 20 and 60 nM) dose-dependently increases cytoplasmic [Ca2+] concentrations with an EC50 value of 92.7 nM in hCaR-HEK293 cells.

Storage Conditions

3 years -20°C powder

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