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ML204

Product Specifications

CAS Number

5465-86-1

Target

TRP Channel

Applications

Neuronal Signaling

Smiles

CC1=CC (=NC2=CC=CC=C12) N3CCCCC3

Molecular Formula

C15H18N2

Additionnal Information

ML204 is a novel, potent, and selective TRPC4 channel inhibitor with apparent IC50 values of about 1 μM in fluorescent intracellular Ca2+ assays and about 3 μM in whole-cell voltage clamp experiments. It exhibits some selectivity within the TRPC subfamily of channels and higher selectivity against other TRP channels and non-TRP channels.

Storage Conditions

2 years -80 in solvent

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