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LRRK2-IN-1

Product Specifications

CAS Number

1234480-84-2

Target

LRRK2

Applications

Autophagy

Smiles

CN1CCN (CC1) C2CCN (CC2) C (=O) C3=CC (=C (C=C3) NC4=NC=C5C (=N4) N (C6=CC=CC=C6C (=O) N5C) C) OC

Molecular Formula

C31H38N8O3

Additionnal Information

LRRK2-IN-1 is a potent and selective LRRK2 inhibitor with IC50 of 6 nM and 13 nM for LRRK2 (G2019S) and LRRK2 (WT), respectively.

Storage Conditions

2 years -80 in solvent

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