Birabresib (OTX015)
Product Specifications
CAS Number
202590-98-5
Synonyms
MK 8628
Target
Epigenetic Reader Domain
Applications
Epigenetics
Smiles
CC1=C (SC2=C1C (=NC (C3=NN=C (N32) C) CC (=O) NC4=CC=C (C=C4) O) C5=CC=C (C=C5) Cl) C
Molecular Formula
C25H22ClN5O2S
Additionnal Information
Birabresib (OTX015, MK 8628) is a potent BET bromodomain inhibitor with EC50 ranging from 10 to 19 nM for BRD2, BRD3, and BRD4 in cell-free assays. Birabresib inhibits the expression of Nuclear receptor binding SET domain protein 3 (NSD3) target genes.
Storage Conditions
2 years -80 in solvent
Frequently Asked Questions
More Discoveries
Explore Other Products
Browse additional items from our catalog
BNC881994-100 1x 100 µL
MMP3 (Marker of Metastasis and Rheumatoid Arthritis) (MMP3/1994R), CF488A conjugate, 0.1mg/mL
Sign In for Pricing
View Details 
![Glucocorticoid Receptor (NR3C1) Mouse Monoclonal Antibody [Clone ID: OTI2C4]](https://cdn.genprice.uk/products/937/68dd18b9061270361e907e77/imageurl/cf806187.webp)
CF806187 100 µg
Glucocorticoid Receptor (NR3C1) Mouse Monoclonal Antibody [Clone ID: OTI2C4]
Sign In for Pricing
View Details 
![Perilipin-1 (PLIN1) Rabbit Monoclonal Antibody [Clone ID: R03-6P-9]](https://cdn.genprice.uk/products/937/68dd1b60061270361ea1223f/imageurl/ta421432.webp)
TA421432 100 µL
Perilipin-1 (PLIN1) Rabbit Monoclonal Antibody [Clone ID: R03-6P-9]
Sign In for Pricing
View Details