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G007-LK

Product Specifications

CAS Number

1380672-07-0

Target

PARP

Applications

DNA Damage/DNA Repair

Smiles

CS (=O) (=O) C1=CN=C (C=C1) C2=NN=C (N2C3=CC=CC=C3Cl) C=CC4=NN=C (O4) C5=CC=C (C=C5) C#N

Molecular Formula

C25H16ClN7O3S

Additionnal Information

G007-LK is a potent and selective tankyrase inhibitor with IC50 of 46 nM and 25 nM for TNKS1/2, respectively.

Storage Conditions

2 years -80 in solvent

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