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ETC-159

Product Specifications

CAS Number

1638250-96-0

Synonyms

ETC-1922159

Target

PORCN

Applications

Cytoskeletal Signaling

Smiles

CN1C2=C (C (=O) N (C1=O) C) N (C=N2) CC (=O) NC3=NN=C (C=C3) C4=CC=CC=C4

Molecular Formula

C19H17N7O3

Additionnal Information

ETC-159 (ETC-1922159) is an orally available, potent porcupine inhibitor with an IC50 of 2.9 nM for inhibiting β-catenin reporter activity in STF3A cells.

Storage Conditions

3 years -20°C powder

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