Elagolix Sodium
Product Specifications
CAS Number
832720-36-2
Synonyms
NBI-56418, ABT-620
Target
GNRH Receptor
Applications
GPCR & G Protein
Smiles
CC1=C (C (=O) N (C (=O) N1CC2=C (C=CC=C2F) C (F) (F) F) CC (C3=CC=CC=C3) NCCCC (=O) [O-]) C4=C (C (=CC=C4) OC) F.[Na+]
Molecular Formula
C32H29F5N3O5.Na
Additionnal Information
Elagolix Soidum (NBI-56418, ABT-620) is a potent, selective, orally active, non-peptide antagonist of the gonadotropin-releasing hormone receptor (GnRHR) with Kd value of 54 pM. Concentration at 10 μM shows no significant activity on ion channels, enzymes, and transporters (inhibition <50%) .
Storage Conditions
2 years -80 in solvent
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