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Tyrphostin AG 879

Product Specifications

CAS Number

148741-30-4

Synonyms

AG 879

Target

HER2

Applications

Protein Tyrosine Kinase

Smiles

CC (C) (C) C1=CC (=CC (=C1O) C (C) (C) C) C=C (C#N) C (=S) N

Molecular Formula

C18H24N2OS

Additionnal Information

Tyrphostin AG 879 potently inhibits HER2/ErbB2 with IC50 of 1 μM, 100- and 500-fold higher selective to ErbB2 than PDGFR and EGFR.

Storage Conditions

2 years -80 in solvent

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