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ZSTK474

Product Specifications

CAS Number

475110-96-4

Target

PI3K

Applications

PI3K/Akt/mTOR

Smiles

C1COCCN1C2=NC (=NC (=N2) N3C4=CC=CC=C4N=C3C (F) F) N5CCOCC5

Molecular Formula

C19H21F2N7O2

Additionnal Information

ZSTK474 inhibits class I PI3K isoforms with IC50 of 37 nM in a cell-free assay, mostly PI3Kδ. Phase1/2.

Storage Conditions

2 years -80 in solvent

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