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BPI-460372

Product Specifications

CAS Number

2762619-63-4

Target

TEAD

Applications

Hippo

Molecular Formula

C18H13F4N5O2

Additionnal Information

BPI‐460372 is an orally available, covalent, irreversible inhibitor of TEAD 1/3/4 that binds to the cysteine residue in the TEAD palmitoylation pocket, preventing palmitoylation and inhibiting TEAD’s transcriptional activity.

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