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BSJ-5-63

Product Specifications

CAS Number

2519823-37-9

Target

CDK

Applications

Cell Cycle

Molecular Formula

C52H74ClN9O6S2

Additionnal Information

BSJ-5-63 is a potent PROTAC degrader of CDK12, CDK7, CDK9. BSJ-5-63 decreases the protein expression of CDK12, CDK7, CDK9, RNAPII, Cyclin K, while also suppressing the mRNA expression of BRCA1 and BRCA2. BSJ-5-63 demonstrates anticancer properties and has the potential for the research of prostate cancer.

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