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Ensifentrine

Product Specifications

CAS Number

1884461-72-6

Synonyms

RPL-554

Target

PDE

Applications

Metabolism

Molecular Formula

C26H31N5O4

Additionnal Information

Ensifentrine (RPL-554) is a first-in-class dual inhibitor of phosphodiesterase 3 (PDE3) and PDE4 with IC50 values of 0.4 nM and 1479 nM, respectively. Ensifentrine also inhibits lipopolysaccharide-induced tumor necrosis factor alpha release from human monocytes in a concentration-dependent manner. Ensifentrine demonstrates bronchoprotective and anti-inflammatory activities and can be used for chronic obstructive pulmonary disease (COPD) research.

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