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SAFit2

Product Specifications

CAS Number

1643125-33-0

Target

FKBP

Applications

Apoptosis

Molecular Formula

C46H62N2O10

Additionnal Information

SAFit2 is a highly potent and selective antagonist of FK506-binding protein 51 (FKBP51) with a Ki of 6 nM. It exhibits anxiolytic and antidepressant-like effects, regulates AKT2-AS160 signaling and metabolic function, and may be useful in research on stress-related disorders and type 2 diabetes.

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