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M4205 (IDRX-42)

Product Specifications

CAS Number

2590556-80-0

Synonyms

IDRX-42

Target

C-Kit

Applications

Protein Tyrosine Kinase

Molecular Formula

C29H32N8O

Additionnal Information

M4205 (IDRX-42) is an oral, selective inhibitor of KIT with broad activity against mutations in KIT exons 11, 13, and 17. It exhibits significant and dose-dependent antitumor activity in the xenograft model of GIST.

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