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Saruparib (AZD5305)

Product Specifications

CAS Number

2589531-76-8

Target

PARP

Applications

DNA Damage/DNA Repair

Molecular Formula

C22H26N6O2

Additionnal Information

Saruparib (AZD5305) is a highly selective and potent inhibitor of PARP1 with an IC50 of 3 nM in wild-type A549 lung cancer cells. AZD5305 shows no or minimal growth inhibitory effects in other cells (IC50s >10μM) .

Storage Conditions

3 years -20°C powder

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