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DTAG-13

Product Specifications

CAS Number

2064175-41-1

Synonyms

FKBP12 PROTAC dTAG-13

Target

FKBP

Applications

Apoptosis

Molecular Formula

C57H68N4O15

Additionnal Information

DTAG-13 (FKBP12 PROTAC dTAG-13) is an ortho-substituted, heterobifunctional selective degrader of FKBP12F36V that effectively engage FKBP12F36V and CRBN leading to rapid and selective CRBN-mediated degradation of FKBP12F36V.It can useful for target validation in the context of drug discovery.

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