Lanraplenib (GS-SYK)
Product Specifications
CAS Number
1800046-95-0
Synonyms
GS-9876
Target
Syk
Applications
Protein Tyrosine Kinase
Smiles
NC1=CN=CC (=N1) C2=C[N]3C=CN=C3C (=N2) NC4=CC=C (C=C4) N5CCN (CC5) C6COC6
Molecular Formula
C23H25N9O
Additionnal Information
Lanraplenib (GS-SYK) is a potent, highly selective and orally active inhibitor of Spleen Tyrosine Kinase (SYK) with IC50 of 9.5 nM. Lanraplenib inhibits SYK activity in platelets via the glycoprotein VI (GPVI) receptor without prolonging bleeding time (BT) in monkeys or humans.
Storage Conditions
3 years -20°C powder
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