BMS-986158
Product Specifications
CAS Number
1800340-40-2
Target
Epigenetic Reader Domain
Applications
Epigenetics
Smiles
C[N]1N=NC (=C1C2=CC3=C (N=C2) C4=C (C=C (C=C4) C (C) (C) O) [N]3C (C5CCOCC5) C6=CC=CC=C6) C
Molecular Formula
C30H33N5O2
Additionnal Information
BMS-986158 is a potent inhibitor of BET with IC50s of 6.6 nM and 5 nM in NCI-H211 small cell lung cancer (SCLC) cells and MDA-MB231 triple negative breast cancer (TNBC) cells, respectively.
Storage Conditions
3 years -20°C powder
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Abi-1 (ABI1, SSH3BP1, Abl interactor 1, Abelson interactor 1, Abi-1, Abl-binding protein 4, AblBP4, Eps8 SH3 domain-binding protein, Eps8-binding protein, Nap1-binding protein, Nap1BP, Spectrin SH3 domain-binding protein 1, e3B1)
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