What is the catalog number for GSK046 (iBET-BD2)?

The catalog number for GSK046 (iBET-BD2) is S9684-100mg.

What sizes are available for GSK046 (iBET-BD2)?

GSK046 (iBET-BD2) is available in the following size(s): 100 mg.

Is GSK046 (iBET-BD2) in stock?

GSK046 (iBET-BD2) is currently made to order / not held in immediate stock. Contact us for lead time.

Who manufactures GSK046 (iBET-BD2)?

GSK046 (iBET-BD2) is manufactured by Bimake.

What is the estimated delivery time for GSK046 (iBET-BD2)?

Estimated delivery time for GSK046 (iBET-BD2) is approximately 15 business day(s), depending on your location.

GSK046 (iBET-BD2)

Product Specifications

CAS Number

2474876-09-8

Target

Epigenetic Reader Domain

Applications

Epigenetics

Smiles

CC (OC1=CC (=CC (=C1NC (C) =O) F) C (=O) NC2CCC (O) CC2) C3=CC=CC=C3

Molecular Formula

C23H27FN2O4

Additionnal Information

GSK046 (iBET-BD2) is a selective and orally active inhibitor of BET (bromodomain and extraterminal domain) with IC50 of 264 nM, 98 nM, 49 nM and 214 nM for BRD2BD2, BRD3BD2, BRD4BD2 and BRDTBD2, respectively. GSK046 exhibits immunomodulatory activity.