GSK778 (iBET-BD1)
Product Specifications
CAS Number
2451862-42-1
Target
Epigenetic Reader Domain
Applications
Epigenetics
Molecular Formula
C30H33N5O3
Additionnal Information
GSK778 (iBET-BD1) is a strong BD1 bromodomain inhibitor of the BET proteins, with IC50 value of 75 nM for BRD2 BD1, 41 nM for BRD3 BD1, 41 nM for BRD4 BD1, and 143 nM for BRDT BD1.
Storage Conditions
3 years -20°C powder
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