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GSK778 (iBET-BD1)

Product Specifications

CAS Number

2451862-42-1

Target

Epigenetic Reader Domain

Applications

Epigenetics

Molecular Formula

C30H33N5O3

Additionnal Information

GSK778 (iBET-BD1) is a strong BD1 bromodomain inhibitor of the BET proteins, with IC50 value of 75 nM for BRD2 BD1, 41 nM for BRD3 BD1, 41 nM for BRD4 BD1, and 143 nM for BRDT BD1.

Storage Conditions

3 years -20°C powder

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