PF-06821497
Product Specifications
CAS Number
1844849-10-0
Target
EZH1/2
Applications
Epigenetics
Smiles
CC1=CC (=C (C (=O) N1) CN2CCC3=C (C=C (C (=C3C2=O) Cl) C (C4COC4) OC) Cl) OC
Molecular Formula
C22H24Cl2N2O5
Additionnal Information
PF-06821497 is a selective and orally active inhibitor of Zeste Homolog 2 (EZH2) with a Ki value <0.1 nM against mutant Y641N EZH2. It exhibits robust tumor growth inhibition.
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