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AS2863619

Product Specifications

CAS Number

2241300-51-4

Target

CDK

Applications

Cell Cycle

Smiles

CC1=NC2=C (N1) C=C (C=C2) N3C4=C (C=NC=C4) N=C3C5=NON=C5N.Cl.Cl

Molecular Formula

C16H14Cl2N8O

Additionnal Information

AS2863619 is a small-molecule cyclin-dependent kinase CDK8/19 inhibitor with IC50 of 0.6099 nM and 4.277 nM, respectively. AS2863619 is a potent Foxp3 inducer in Tconv cells.

Storage Conditions

3 years -20°C powder

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